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Non-sedating H1 antihistamine

Levocetirizine hydrochloride

Brand names: Xyzal

Adult dose

Dose: 5mg PO OD
Route: PO
Frequency: OD

Paediatric dose

Route: PO
Frequency: OD
Age bands
  • 24–72m: 1.25mg BD
  • 72–144m: 2.5mg BD or 5mg OD

Dose adjustments

Renal

CrCl 30–50: 5mg every other day; <10: avoid

Clinical pearls

  • Active enantiomer of cetirizine — slightly cleaner sedation profile
  • Allergic rhinitis, urticaria

Contraindications

  • Severe renal impairment (CrCl <10)

Side effects

  • Drowsiness (less than cetirizine)
  • Headache
  • Dry mouth

Interactions

  • CNS depressants

Reference: BNFc; BNF; BSACI rhinitis/urticaria guidelines; https://bnf.nice.org.uk/drugs/levocetirizine-hydrochloride/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.