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Fibrate / PPAR-α agonist

Ciprofibrate

Brand names: Modalim

Adult dose

Dose: 100mg OD
Route: PO
Frequency: OD

Clinical pearls

  • Used for severe hypertriglyceridaemia not responding to lifestyle/statin
  • Check CK before starting and if symptoms

Contraindications

  • Severe renal impairment (CrCl <60)
  • Hepatic impairment
  • Gallbladder disease
  • Pregnancy/breastfeeding

Side effects

  • Myopathy / rhabdomyolysis
  • GI upset
  • Headache
  • Cholelithiasis
  • Erectile dysfunction

Interactions

  • Statins — myopathy risk (avoid combination if possible)
  • Warfarin — INR rise
  • Ciclosporin — renal toxicity

Monitoring

  • LFTs
  • Lipids
  • CK if symptoms
  • U&E

Reference: BNF; NICE CG181; https://bnf.nice.org.uk/drugs/ciprofibrate/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.