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Phosphodiesterase-3 inhibitor (inotrope/vasodilator)

Enoximone

Brand names: Perfan

Adult dose

Dose: Loading 0.5–1mg/kg IV slowly; infusion 5–20 micrograms/kg/min titrated
Route: IV
Frequency: Continuous infusion

Clinical pearls

  • Short-term decompensated HF / cardiogenic shock — ICU/CCU only
  • Largely superseded by milrinone in many UK centres
  • ESC HF acute decompensation guidance — inotropes for cardiogenic shock with hypoperfusion

Contraindications

  • Severe outflow obstruction (HOCM, severe AS)
  • Hypovolaemia (correct first)
  • Hypersensitivity

Side effects

  • Hypotension
  • Arrhythmias (ventricular and supraventricular)
  • Thrombocytopenia
  • Headache
  • Nausea

Interactions

  • Other inotropes/vasodilators
  • QT-prolonging drugs

Monitoring

  • Continuous ECG
  • BP
  • Cardiac output
  • Platelets
  • Electrolytes

Reference: BNF; ESC acute HF guidelines; AAGBI ICU; SmPC; https://bnf.nice.org.uk/drugs/enoximone/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.