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α1-adrenergic antagonist

Terazosin

Brand names: Hytrin

Adult dose

Dose: BPH/HTN: initial 1mg ON, titrate weekly to 5–10mg OD
Route: PO
Frequency: OD

Clinical pearls

  • BPH, resistant hypertension
  • First dose at bedtime to mitigate hypotension

Contraindications

  • Postural hypotension
  • Hypersensitivity

Side effects

  • First-dose hypotension
  • Dizziness
  • Asthenia
  • Nasal congestion
  • Priapism (rare)
  • IFIS

Interactions

  • Other antihypertensives
  • PDE5 inhibitors
  • α-blockers

Reference: BNF; NICE NG106; https://bnf.nice.org.uk/drugs/terazosin/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.