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K-sparing diuretic (ENaC blocker)

Triamterene

Brand names: Dytac

Adult dose

Dose: 150–250mg PO/day in divided doses
Route: PO
Frequency: OD-BD

Dose adjustments

Renal

Avoid if eGFR <30

Clinical pearls

  • Adjunct to thiazides/loop in oedema; rarely used alone
  • Take with food

Contraindications

  • Hyperkalaemia
  • Severe renal impairment
  • Concurrent K-sparing diuretic / K supplements
  • Anuria
  • Severe hepatic impairment

Side effects

  • Hyperkalaemia
  • GI upset
  • Megaloblastic anaemia (folate antagonism)
  • Renal stones (rare)
  • Blue urine fluorescence

Interactions

  • ACEi/ARB
  • Lithium
  • NSAIDs
  • K supplements

Monitoring

  • U&E
  • K+

Reference: BNF; NICE; https://bnf.nice.org.uk/drugs/triamterene/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.