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JAK3/TEC kinase inhibitor

Ritlecitinib

Brand names: Litfulo

Adult dose

Dose: 50mg PO OD
Route: PO
Frequency: OD

Clinical pearls

  • Severe alopecia areata in adults/adolescents ≥12y per NICE TA958
  • Pre-treatment screening: TB, hepatitis, varicella, malignancy

Contraindications

  • Active serious infection
  • Active malignancy
  • Severe hepatic impairment
  • Pregnancy
  • Hypersensitivity

Side effects

  • Infections (incl. herpes zoster, TB reactivation)
  • MACE
  • Malignancy
  • VTE
  • Cytopenias
  • Hepatotoxicity
  • Folliculitis
  • Headache

Interactions

  • Live vaccines
  • Strong CYP3A4 modulators
  • Other immunosuppressives

Monitoring

  • FBC
  • Lipids
  • LFTs
  • Infections

Reference: BNF; NICE TA958; MHRA JAKi class; SmPC; https://bnf.nice.org.uk/drugs/ritlecitinib/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.