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Sulfonylurea (2nd generation)

Glipizide

Brand names: Glibenese, Minodiab

Adult dose

Dose: 2.5–5mg OD before breakfast; usual range 2.5–20mg/day; max 20mg/day (in divided doses if >15mg)
Route: PO
Frequency: OD or BD

Clinical pearls

  • Less commonly used than gliclazide in UK
  • Take 30 min before food

Contraindications

  • Type 1 diabetes
  • DKA
  • Severe hepatic/renal impairment
  • Pregnancy/breastfeeding
  • Porphyria

Side effects

  • Hypoglycaemia
  • Weight gain
  • GI upset
  • Hyponatraemia
  • Cholestatic jaundice (rare)

Interactions

  • Other hypoglycaemics
  • β-blockers (mask hypoglycaemia)
  • Alcohol
  • CYP2C9 inhibitors

Monitoring

  • HbA1c
  • Hypoglycaemia symptoms

Reference: BNF; NICE NG28; https://bnf.nice.org.uk/drugs/glipizide/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.