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Carbapenem + β-lactamase inhibitor

Imipenem with cilastatin and relebactam

Brand names: Recarbrio

Adult dose

Dose: 1.25g IV every 6h (refer to BNF for renal dose)
Route: IV
Frequency: q6h

Dose adjustments

Renal

Mandatory — refer to BNF

Clinical pearls

  • Activity against KPC-producing carbapenem-resistant Enterobacterales; specialist micro/ID input

Contraindications

  • Hypersensitivity

Side effects

  • As imipenem
  • Diarrhoea
  • Hepatotoxicity

Interactions

  • Valproate (avoid)
  • Other carbapenem interactions

Monitoring

  • U&E
  • LFTs
  • FBC

Reference: BNF; SmPC; https://bnf.nice.org.uk/drugs/imipenem-with-cilastatin-and-relebactam/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.