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Fumaric acid ester (prodrug of monomethyl fumarate)

Diroximel fumarate

Brand names: Vumerity

Adult dose

Dose: Start 231mg BD for 7 days, then 462mg BD
Route: Oral
Frequency: BD

Clinical pearls

  • Relapsing-remitting MS — alternative to dimethyl fumarate with improved GI tolerability
  • NICE TA evaluation; ABN MS-DMT guidance
  • Same active metabolite (MMF) as dimethyl fumarate

Contraindications

  • Severe lymphopaenia
  • Active serious infection
  • Severe renal/hepatic impairment
  • Hypersensitivity

Side effects

  • Flushing (less than dimethyl fumarate)
  • GI events (less than dimethyl fumarate)
  • Lymphopaenia
  • PML (rare, JCV)
  • Hepatotoxicity

Interactions

  • Immunosuppressives
  • Live vaccines

Monitoring

  • FBC (lymphocytes)
  • LFTs
  • Renal
  • JCV antibody if prolonged lymphopaenia

Reference: BNF; NICE TA evaluation; ABN MS-DMT; SmPC; https://bnf.nice.org.uk/drugs/diroximel-fumarate/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.