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Barbiturate-derived antiepileptic

Primidone

Brand names: Mysoline

Adult dose

Dose: Initial 125mg ON, increase by 125mg every 3 days; usual 0.5–1.5g/day in 2 divided doses. Essential tremor: 25–250mg ON
Route: PO
Frequency: BD or ON

Clinical pearls

  • Essential tremor (2nd-line after propranolol); generalised tonic-clonic seizures
  • Largely superseded; metabolised to phenobarbital

Contraindications

  • Acute porphyria
  • Severe respiratory disease
  • Hypersensitivity

Side effects

  • Sedation
  • Ataxia
  • Megaloblastic anaemia
  • Osteomalacia
  • Connective tissue disorders
  • Withdrawal seizures

Interactions

  • Many — strong enzyme inducer
  • Hormonal contraceptives
  • Anticoagulants
  • Many AEDs

Monitoring

  • FBC
  • LFTs
  • Drug levels (rarely)

Reference: BNF; NICE NG217; https://bnf.nice.org.uk/drugs/primidone/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.