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Enzymatic Debriding Agent Pregnancy: C

Collagenase (Wound Debridement)

Brand names: Santyl, Iruxol Mono

Adult dose

Dose: Apply once daily to wound bed after cleansing; cover with moist dressing
Route: topical
Frequency: once daily
Max: Topical use only
Clostridium histolyticum collagenase — selectively digests collagen in necrotic tissue; preserve surrounding healthy tissue; discontinue when wound clean

Paediatric dose

Route: topical
Frequency: once daily
Concentration: 250 units/g ointment /ml
Limited paediatric data; used in specialist burns/wound care settings for debridement; same principles as adults

Dose adjustments

Renal

Not applicable (topical)

Hepatic

Not applicable

Clinical pearls

  • Do NOT use with silver-containing dressings or antiseptics — inactivates the enzyme
  • Iruxol Mono preferred over Iruxol (no neomycin — lower sensitisation risk)
  • Best evidence for partial thickness burns and pressure ulcers — promotes healing by removing necrotic tissue without damaging granulation tissue

Contraindications

  • Hypersensitivity to collagenase or Clostridium components

Side effects

  • Local pain/burning on application
  • Contact dermatitis
  • Potential for increased wound exudate

Interactions

  • Heavy metal ions (mercury, silver — inactivate enzyme)
  • Hydrogen peroxide (inactivates collagenase)
  • Povidone-iodine (inactivates enzyme — do NOT use concurrently)

Monitoring

  • Wound healing progress
  • Signs of local hypersensitivity
  • Wound bed preparation assessment

Reference: BNFc; BNF 86; BBA wound care guidelines; Wounds UK best practice. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.