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ACE inhibitor

Lisinopril

Brand names: Zestril, Carace

Adult dose

Dose: Initial 2.5–10mg OD; usual maintenance 10–40mg OD; max 80mg OD
Route: PO
Frequency: OD

Dose adjustments

Renal

Reduce in CKD; close U&E monitoring

Clinical pearls

  • Hypertension, heart failure, post-MI, diabetic nephropathy
  • Once-daily, no metabolite, useful in hepatic impairment

Contraindications

  • History of angioedema
  • Bilateral renal artery stenosis
  • Pregnancy
  • Concurrent sacubitril/valsartan
  • Concurrent aliskiren in diabetes/CKD

Side effects

  • Cough
  • Hyperkalaemia
  • Renal impairment
  • Angioedema
  • First-dose hypotension
  • Rash

Interactions

  • NSAIDs
  • Potassium-sparing diuretics
  • Lithium
  • Sacubitril/valsartan (avoid concurrent)

Monitoring

  • U&E (1–2 weeks after start, with dose changes)
  • BP

Reference: BNF; NICE NG136/NG106; https://bnf.nice.org.uk/drugs/lisinopril/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.