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Bradykinin B2 receptor antagonist

Icatibant

Brand names: Firazyr

Adult dose

Dose: 30mg SC; may repeat every 6h up to 3 doses/24h
Route: SC
Frequency: per attack

Clinical pearls

  • Acute attacks of hereditary angioedema (C1-INH deficiency) in adults and adolescents ≥2y
  • Self-administration after training

Contraindications

  • Acute coronary syndrome (caution — may worsen ischaemia)
  • Recent stroke

Side effects

  • Injection site reactions (very common)
  • Dizziness
  • Pyrexia

Interactions

  • ACE inhibitors (theoretical antagonism)

Reference: BNF; NICE TA484; SmPC; https://bnf.nice.org.uk/drugs/icatibant/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.