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H1 antihistamine (topical)

Azelastine hydrochloride

Brand names: Rhinolast, Optilast, Dymista (with fluticasone)

Adult dose

Dose: Nasal: 1 spray each nostril BD; Eye: 1 drop BD
Route: Intranasal / Ophthalmic
Frequency: BD

Clinical pearls

  • BSACI / NICE CKS Allergic rhinitis: intranasal antihistamine option (with or without intranasal corticosteroid)
  • RCOphth allergic conjunctivitis
  • Dymista combination first-line for moderate-severe persistent rhinitis

Contraindications

  • Hypersensitivity

Side effects

  • Bitter taste
  • Local irritation
  • Headache
  • Drowsiness (rare)
  • Application-site burning

Interactions

  • Minimal systemic

Monitoring

  • Symptom relief

Reference: BNF; BSACI; NICE CKS Allergic rhinitis; RCOphth; https://bnf.nice.org.uk/drugs/azelastine-hydrochloride/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.