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Cap-dependent endonuclease inhibitor (antiviral)

Baloxavir marboxil

Brand names: Xofluza

Adult dose

Dose: 40mg PO single dose (≥80kg: 80mg)
Route: Oral
Frequency: Single dose

Clinical pearls

  • NICE NG34 / TA evaluation: alternative to oseltamivir for influenza A/B treatment within 48h
  • UKHSA influenza guidance
  • Single-dose convenience but resistance signal monitored

Contraindications

  • Hypersensitivity

Side effects

  • Diarrhoea
  • Headache
  • Hypersensitivity
  • Bronchitis
  • Sinusitis

Interactions

  • Polyvalent cation products (separate by 2h)

Monitoring

  • Symptom resolution

Reference: BNF; NICE NG34; UKHSA influenza; SmPC; https://bnf.nice.org.uk/drugs/baloxavir-marboxil/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.