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NRTI (antiretroviral)

Emtricitabine

Brand names: Emtriva

Adult dose

Dose: 200mg OD
Route: Oral
Frequency: OD

Clinical pearls

  • Component of multiple HIV combination therapies
  • BHIVA HIV guidelines
  • Active against HBV — avoid abrupt discontinuation in HBV co-infection (flare risk)

Contraindications

  • Hypersensitivity

Side effects

  • Hyperpigmentation (palms/soles)
  • Headache
  • GI upset
  • Lactic acidosis (class)
  • HBV reactivation if discontinued in HBV co-infection

Interactions

  • Adefovir/lamivudine (avoid combination)

Monitoring

  • FBC
  • Renal function
  • Viral load
  • HBV serology

Reference: BNF; BHIVA HIV guidelines; EACS guidelines; https://bnf.nice.org.uk/drugs/emtricitabine/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.