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Carbapenem antibiotic

Imipenem with cilastatin

Brand names: Primaxin

Adult dose

Dose: 500mg–1g IV every 6–8h (max 4g/day)
Route: IV
Frequency: q6-8h

Dose adjustments

Renal

Mandatory — refer to BNF

Clinical pearls

  • Severe gram-negative infections incl. ESBL; meropenem usually preferred (lower seizure risk)
  • Cilastatin protects against renal dehydropeptidase

Contraindications

  • Hypersensitivity to carbapenems
  • Severe penicillin allergy (cross-reactivity)

Side effects

  • Seizures (highest seizure risk among carbapenems)
  • Nausea
  • Diarrhoea
  • C. difficile
  • Eosinophilia
  • Hypersensitivity

Interactions

  • Valproate (avoid — markedly reduced valproate levels)
  • Probenecid
  • Ganciclovir (seizures)

Monitoring

  • U&E
  • FBC
  • Neurological exam

Reference: BNF; UK AMR guidance; https://bnf.nice.org.uk/drugs/imipenem-with-cilastatin/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.