ClinCalc Pro
Menu
Oxazolidinone antibiotic

Linezolid

Brand names: Zyvox

Adult dose

Dose: 600mg IV/PO every 12h for 10–28 days (per indication)
Route: IV/PO
Frequency: BD

Clinical pearls

  • MRSA, VRE, complicated SSTI, MDR-TB
  • Restricted use — micro/AMR approval; FBC weekly

Contraindications

  • Concurrent MAOI / SSRI / SNRI / TCA / triptan / pethidine (serotonin syndrome — avoid unless monitored)
  • Uncontrolled hypertension
  • Phaeochromocytoma
  • Carcinoid
  • Severe untreated thyroid disease
  • Pregnancy/breastfeeding (relative)

Side effects

  • Thrombocytopenia / cytopenias (limit course ≤28 days)
  • Lactic acidosis
  • Optic neuropathy / peripheral neuropathy (prolonged use)
  • Serotonin syndrome with serotonergic drugs
  • GI upset

Interactions

  • Serotonergic drugs — major
  • Tyramine-rich foods
  • Sympathomimetics
  • Adrenaline / dopamine (raised pressor effect)

Monitoring

  • FBC weekly
  • Lactate if symptoms
  • Visual symptoms
  • Mental state for serotonin syndrome

Reference: BNF; NICE CKS; UK AMR guidance; https://bnf.nice.org.uk/drugs/linezolid/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.