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Sulfonamide antibiotic

Sulfadiazine

Adult dose

Dose: Toxoplasmosis: 1–1.5g PO QDS with pyrimethamine + folinic acid (specialist)
Route: PO
Frequency: QDS

Clinical pearls

  • Toxoplasmosis (with pyrimethamine + folinic acid)
  • Always co-prescribe folinic acid

Contraindications

  • Sulfonamide hypersensitivity
  • Severe renal/hepatic impairment
  • Porphyria
  • Pregnancy/breastfeeding (caution)
  • G6PD deficiency

Side effects

  • SJS/TEN
  • Hepatotoxicity
  • Cytopenias
  • Crystalluria (maintain hydration)
  • Hypersensitivity
  • Photosensitivity

Interactions

  • Methotrexate
  • Warfarin
  • Sulfonylureas
  • Phenytoin

Monitoring

  • FBC
  • U&E
  • LFTs
  • Hydration

Reference: BNF; BHIVA; SmPC; https://bnf.nice.org.uk/drugs/sulfadiazine/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.