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Tricyclic antidepressant

Imipramine hydrochloride

Adult dose

Dose: Depression: 75mg/day initial, increase to 150–200mg/day. Nocturnal enuresis (≥7y): 25–50mg nocte (max 75mg)
Route: PO
Frequency: OD or divided

Clinical pearls

  • Nocturnal enuresis when non-pharmacological + desmopressin failed (specialist)

Contraindications

  • Recent MI
  • Arrhythmia
  • Mania
  • Severe hepatic impairment
  • Concurrent MAOI

Side effects

  • Anticholinergic
  • Sedation
  • Cardiac conduction delay
  • Lowered seizure threshold
  • Weight gain
  • Urinary retention

Interactions

  • MAOIs (avoid)
  • SSRIs
  • QT-prolonging drugs
  • CYP2D6 inhibitors

Monitoring

  • BP
  • ECG if cardiac risk

Reference: BNF; NICE NG28 (children); https://bnf.nice.org.uk/drugs/imipramine-hydrochloride/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.