ClinCalc Pro
Menu
Antihistamine (Non-Sedating) Pregnancy: B — generally considered safe

Cetirizine

Brand names: Zirtek, Piriteze

Adult dose

Dose: 10mg once daily
Route: Oral
Frequency: Once daily
Renal impairment: eGFR 30–50 → 5mg OD; eGFR <30 → 5mg every other day.

Paediatric dose

Route: Oral
Frequency: Once or twice daily
6–12 years: 5mg BD or 10mg OD. 2–6 years: 2.5mg BD or 5mg OD. Under 2 years: not recommended.

Clinical pearls

  • Preferred over chlorphenamine (first-generation) for daytime use — less sedating
  • For chronic urticaria: can dose up to 20–40mg/day (unlicensed) under specialist guidance
  • Levocetirizine (active enantiomer) — half the dose for same effect (5mg OD)
  • Non-sedating antihistamines do not treat anaphylaxis — use adrenaline first

Contraindications

  • Severe renal impairment (eGFR <10)
  • Hypersensitivity to hydroxyzine

Side effects

  • Drowsiness (less than first-generation)
  • Dry mouth
  • Headache
  • Urinary retention (rare)

Interactions

  • Alcohol — increased CNS depression
  • Theophylline — slightly reduces cetirizine clearance

Monitoring

  • Symptom response
  • No routine monitoring required

Reference: BNFc; BNF; EAACI/GA²LEN/EDF Guidelines on Urticaria 2022. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.