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Centrally-acting non-opioid analgesic

Nefopam hydrochloride

Brand names: Acupan

Adult dose

Dose: 30–90mg TDS PO. IM 20mg every 6h. IV 20mg every 4h
Route: PO/IM/IV
Frequency: TDS-QDS

Clinical pearls

  • Moderate non-opioid analgesia
  • Pink-coloured urine harmless

Contraindications

  • Convulsive disorders
  • Concurrent MAOI
  • Hypersensitivity
  • Children <12

Side effects

  • Anticholinergic effects
  • Sweating
  • Nausea
  • Insomnia
  • Tachycardia
  • Confusion in elderly

Interactions

  • MAOIs
  • TCAs
  • Anticholinergic drugs

Reference: BNF; https://bnf.nice.org.uk/drugs/nefopam-hydrochloride/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.