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Tetracycline antibiotic

Oxytetracycline

Brand names: Imperacin

Adult dose

Dose: 250–500mg QDS on empty stomach
Route: PO
Frequency: QDS

Clinical pearls

  • Acne, rosacea (lower preference than doxycycline/lymecycline)
  • Take on empty stomach with adequate water

Contraindications

  • Pregnancy/breastfeeding
  • Children <12
  • Severe renal impairment
  • Acute porphyria
  • SLE (caution)

Side effects

  • GI upset
  • Photosensitivity
  • Tooth discolouration (children)
  • Hepatotoxicity
  • Benign intracranial hypertension
  • Oesophageal ulceration

Interactions

  • Antacids/iron/calcium/dairy (chelation; separate by 2h)
  • Warfarin (raised INR)
  • Methotrexate (raised levels)

Monitoring

  • LFTs in prolonged use

Reference: BNF; NICE NG198 acne; https://bnf.nice.org.uk/drugs/oxytetracycline/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.