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Antimuscarinic (M3-selective)

Solifenacin succinate

Brand names: Vesicare

Adult dose

Dose: 5mg PO OD; may increase to 10mg OD
Route: PO
Frequency: OD

Dose adjustments

Renal

Max 5mg if eGFR <30

Clinical pearls

  • Overactive bladder
  • Mirabegron preferred in older adults to reduce cognitive risk

Contraindications

  • Urinary retention
  • GI obstruction
  • Glaucoma
  • Myasthenia gravis
  • Severe ulcerative colitis
  • Toxic megacolon
  • Severe hepatic impairment

Side effects

  • Dry mouth
  • Constipation
  • Blurred vision
  • QT prolongation
  • Anticholinergic burden

Interactions

  • Strong CYP3A4 inhibitors (max 5mg)
  • QT-prolonging drugs
  • Other antimuscarinics

Monitoring

  • Symptoms
  • Anticholinergic burden

Reference: BNF; NICE NG123; https://bnf.nice.org.uk/drugs/solifenacin-succinate/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.