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Fibrate

Gemfibrozil

Brand names: Lopid

Adult dose

Dose: 1.2g/day in 2 divided doses (max 1.5g/day)
Route: PO
Frequency: BD

Clinical pearls

  • Severe hypertriglyceridaemia where fenofibrate not suitable; rarely used now
  • Major drug-interaction risk: avoid with statins

Contraindications

  • Severe hepatic/renal impairment
  • Gallbladder disease
  • Concurrent statins (rhabdomyolysis — avoid combination, particularly with simvastatin/atorvastatin/pravastatin)
  • Concurrent repaglinide/dasabuvir

Side effects

  • Myopathy/rhabdomyolysis
  • GI upset
  • Cholelithiasis

Interactions

  • Statins — AVOID combination
  • Repaglinide (severe hypoglycaemia)
  • Warfarin (raised INR)

Monitoring

  • Lipids
  • LFTs
  • CK if symptoms

Reference: BNF; NICE CG181; https://bnf.nice.org.uk/drugs/gemfibrozil/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.