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Organic nitrate

Isosorbide mononitrate

Brand names: Imdur, Monomil, Ismo, Elantan

Adult dose

Dose: PO immediate-release 20–40mg BD asymmetric dosing (nitrate-free interval). Modified-release 60–120mg OD
Route: PO
Frequency: OD-BD

Clinical pearls

  • Asymmetric dosing (e.g. 8am + 2pm IR) provides nitrate-free interval to prevent tolerance

Contraindications

  • Marked hypotension
  • Concurrent PDE-5 inhibitors
  • Severe aortic stenosis

Side effects

  • Headache
  • Flushing
  • Hypotension
  • Tachycardia

Interactions

  • PDE-5 inhibitors
  • Riociguat

Monitoring

  • BP

Reference: BNF; NICE NG185; https://bnf.nice.org.uk/drugs/isosorbide-mononitrate/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.