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Fifth-generation cephalosporin (anti-MRSA)

Ceftaroline fosamil

Brand names: Zinforo

Adult dose

Dose: 600mg IV q12h
Route: IV
Frequency: q12h

Clinical pearls

  • BSAC: MRSA cover within cephalosporin class
  • ABSSSI / community-acquired pneumonia (UKHSA AMR — restricted)
  • Off-label for MRSA bacteraemia / endocarditis (specialist microbiology)

Contraindications

  • Severe beta-lactam hypersensitivity

Side effects

  • GI upset
  • Hypersensitivity
  • C. difficile
  • Eosinophilia
  • Direct Coombs positivity

Interactions

  • Limited

Monitoring

  • Renal function
  • C. diff
  • Coombs

Reference: BNF; BSAC; UKHSA AMR; SmPC; https://bnf.nice.org.uk/drugs/ceftaroline-fosamil/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.