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CDK4/6 inhibitor

Abemaciclib [Specialist drug]

Brand names: Verzenios

Adult dose

Dose: Specialist (typically 150 mg BD with endocrine therapy; 200 mg BD monotherapy)
Route: Oral
Frequency: Per SACT/SmPC

Clinical pearls

  • Refer to BNF/SmPC and SACT protocol; do not initiate outside oncology MDT
  • Loperamide on hand for diarrhoea

Contraindications

  • Severe hepatic impairment (per SmPC)

Side effects

  • Diarrhoea (often early/severe)
  • Neutropenia
  • Fatigue
  • VTE
  • ILD

Interactions

  • Strong CYP3A inhibitors/inducers
  • Grapefruit juice

Monitoring

  • FBC, LFTs
  • VTE/ILD symptoms

Reference: BNF; NICE TA563/TA810; ESMO; SmPC Verzenios. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.