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Hydrazine alkylating cytotoxic

Procarbazine (Specialist drug)

Adult dose

Dose: Specialist initiation only — refer to BNF/SmPC
Route: PO
Frequency: per protocol

Clinical pearls

  • Hodgkin lymphoma (BEACOPP/escalated regimens); high-grade glioma (PCV)
  • Specialist haem-onc; avoid tyramine

Contraindications

  • Severe myelosuppression
  • Severe hepatic/renal impairment
  • Pregnancy

Side effects

  • Severe myelosuppression
  • Nausea/vomiting
  • Hypersensitivity
  • MAOI-like effects (avoid tyramine)
  • Pulmonary fibrosis
  • Secondary malignancy

Interactions

  • Tyramine-rich foods
  • Sympathomimetics
  • TCAs
  • Alcohol (disulfiram-like)
  • Other MAOIs

Monitoring

  • FBC
  • LFTs

Reference: BNF; SmPC; https://bnf.nice.org.uk/drugs/procarbazine-specialist-drug/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.