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Class Ic antiarrhythmic

Propafenone hydrochloride

Brand names: Arythmol

Adult dose

Dose: 150mg PO TDS initially, increase to 300mg TDS (max 900mg/day). 'Pill in pocket' for AF: 450–600mg single
Route: PO
Frequency: TDS

Clinical pearls

  • Paroxysmal AF (no structural heart disease) — 'pill in pocket'
  • Specialist initiation; ECG mandatory

Contraindications

  • Heart failure
  • Cardiogenic shock
  • Severe bradycardia/AV block
  • Recent MI
  • Structural heart disease
  • Severe COPD
  • Myasthenia gravis

Side effects

  • Pro-arrhythmia
  • Bradycardia
  • Heart block
  • Bronchospasm
  • Metallic taste
  • Hepatotoxicity

Interactions

  • Digoxin
  • Warfarin
  • β-blockers
  • Strong CYP2D6 inhibitors
  • QT-prolonging drugs

Monitoring

  • ECG
  • LFTs
  • FBC

Reference: BNF; NICE NG196; ESC; https://bnf.nice.org.uk/drugs/propafenone-hydrochloride/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.