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Tetracycline antibiotic / off-label SIADH treatment

Demeclocycline hydrochloride

Brand names: Ledermycin

Adult dose

Dose: SIADH (off-label): 600–1,200mg/day in divided doses
Route: Oral
Frequency: BD–QDS

Clinical pearls

  • Renal AVP-V2 antagonist effect — used in chronic SIADH unresponsive to fluid restriction
  • Society for Endocrinology / RCP hyponatraemia guidance — vaptans (tolvaptan) generally preferred where available
  • Specialist endocrinology supervision

Contraindications

  • Pregnancy
  • Children <12
  • Severe hepatic/renal impairment
  • Hypersensitivity

Side effects

  • Diabetes insipidus (intended in SIADH; unintended in infection use)
  • Photosensitivity
  • GI upset
  • Tooth discolouration in young children
  • Pseudotumor cerebri

Interactions

  • Cation-containing products (chelation)
  • Warfarin
  • Penicillins (antagonism)

Monitoring

  • Sodium
  • Renal function
  • LFTs
  • Urine output

Reference: BNF; Society for Endocrinology hyponatraemia guidance; RCP; https://bnf.nice.org.uk/drugs/demeclocycline-hydrochloride/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.