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siRNA targeting transthyretin (TTR)

Patisiran

Brand names: Onpattro

Adult dose

Dose: 300 micrograms/kg IV every 3 weeks (max 30mg)
Route: IV
Frequency: q3w

Clinical pearls

  • Hereditary transthyretin amyloidosis with polyneuropathy; specialist amyloid centre
  • Vitamin A 2500 IU/day required

Contraindications

  • Hypersensitivity

Side effects

  • Infusion reactions
  • Vitamin A deficiency
  • Headache
  • Atrial fibrillation

Interactions

  • Pre-medicate with steroid + antihistamine + paracetamol

Monitoring

  • Cardiac function
  • Vitamin A levels

Reference: BNF; NICE HST10; SmPC; https://bnf.nice.org.uk/drugs/patisiran/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.