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Carbonic anhydrase inhibitor + beta-blocker (combination eye drops)

Dorzolamide with timolol

Brand names: Cosopt

Adult dose

Dose: 1 drop into affected eye(s) BD
Route: Ophthalmic
Frequency: BD

Clinical pearls

  • NICE NG81 glaucoma: combination eye drops when monotherapy inadequate; reduces drop burden and improves adherence
  • RCOphth glaucoma pathway
  • Punctal occlusion 1 minute after instillation reduces systemic absorption

Contraindications

  • Severe asthma
  • Severe COPD
  • Bradyarrhythmia / heart block
  • Heart failure (timolol)
  • Severe renal impairment (dorzolamide)
  • Sulfonamide hypersensitivity
  • Hypersensitivity

Side effects

  • Ocular: burning, taste disturbance, blurred vision, conjunctival injection
  • Systemic: bronchospasm, bradycardia, depression, hypoglycaemia masking, fatigue

Interactions

  • Systemic beta-blockers (additive)
  • Verapamil/diltiazem (bradycardia)
  • Insulin/oral hypoglycaemics (hypoglycaemia mask)
  • Other oral CAIs

Monitoring

  • IOP
  • Visual fields
  • HR/BP if cardiovascular risk
  • Asthma symptoms

Reference: BNF; NICE NG81; RCOphth; https://bnf.nice.org.uk/drugs/dorzolamide-with-timolol/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.