ClinCalc Pro
Menu
BTK inhibitor

Ibrutinib (Specialist drug)

Brand names: Imbruvica

Adult dose

Dose: Specialist initiation only — refer to BNF/SmPC
Route: PO
Frequency: OD

Clinical pearls

  • CLL, mantle cell lymphoma, Waldenström's macroglobulinaemia

Contraindications

  • Concurrent strong CYP3A4 inducers/inhibitors without adjustment

Side effects

  • Bleeding
  • Atrial fibrillation
  • Hypertension
  • Infections (esp. opportunistic)
  • Cytopenias
  • Tumour lysis syndrome

Interactions

  • Strong CYP3A4 modulators
  • Anticoagulants/antiplatelets (bleeding)

Monitoring

  • FBC
  • BP
  • ECG
  • Bleeding

Reference: BNF; NICE TA429/TA491; SmPC; https://bnf.nice.org.uk/drugs/ibrutinib-specialist-drug/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.