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Antimuscarinic (overactive bladder)

Fesoterodine fumarate

Brand names: Toviaz

Adult dose

Dose: 4mg OD initially, increase to 8mg if needed
Route: PO
Frequency: OD

Dose adjustments

Renal

Severe renal impairment: max 4mg OD

Clinical pearls

  • Alternative to oxybutynin/solifenacin
  • Mirabegron preferred in older adults to reduce anticholinergic burden

Contraindications

  • Urinary retention
  • Gastric retention
  • Uncontrolled angle-closure glaucoma
  • Myasthenia gravis
  • Severe hepatic impairment

Side effects

  • Dry mouth
  • Constipation
  • Dyspepsia
  • Urinary retention

Interactions

  • Strong CYP3A4 inhibitors (max 4mg)
  • Other antimuscarinics — additive load

Reference: BNF; NICE NG123; https://bnf.nice.org.uk/drugs/fesoterodine-fumarate/. Verify against your local formulary and the latest BNF before prescribing.

Related

Curated clinical cross-links plus same-class fallbacks.